Organic letters

Direct Intermolecular Aniline Ortho-Arylation via Benzyne Intermediates

T Truong, O Daugulis

文献索引：Organic Letters, , vol. 14, # 23 p. 5964 - 5967

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被引用次数: 11

摘要

... Organic Letters. ... a Total volume of solvent 0.9 mL, 0.25 mmol scale, 24 h; 12 h for entry 5. See the Supporting Information for details. b ... is arylated at the 7-position in good yield (entry 2). Unsubstituted anilines can be selectively and efficiently monoarylated (entries 6–14). ...