RSC Advances

A one-pot process for palladium catalyzed direct C–H acylation of anilines in water using a removable ortho directing group

F Szabó, D Simkó, Z Novák

文献索引：Szabo, Fruzsina; Simko, Daniel; Novak, Zoltan RSC Advances, 2014 , vol. 4, # 8 p. 3883 - 3886

被引用次数: 9

摘要

A new mild, practical method for the synthesis of aminobenzophenone derivatives through a three step one-pot reaction sequence involving acylation of anilines, palladium catalyzed cross-dehydrogenative coupling of the formed anilides and the hydrolytic cleavage is reported. The full reaction sequence was performed under aqueous conditions.

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