Organic Letters

γ-Turn mimicry with benzodiazepinones and pyrrolobenzodiazepinones synthesized from a common amino ketone intermediate

AA Dörr, WD Lubell

文献索引：Perez-Picaso, Lemuel; Escalante, Jaime; Olivo, Horacio F.; Rios, Maria Yolanda Molecules, 2009 , vol. 14, # 8 p. 2836 - 2849

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被引用次数: 2

摘要

... Volume: Page: ... by Boc group removal with HCl gas in DCM, free-basing with triethylamine in the presence of 4 Å molecular sieves in ... and medicinal chemistry because of the importance of γ-turns in peptide biology(33) and the activity of related small molecules. ...

~92%

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