Diastereoselective synthesis, activity and chiral stability of cyclic alkoxyketone inhibitors of cathepsin K

…, AD Gribble, RJ Ife, N Stevens, J Witherington

文献索引：Fenwick, Ashley E.; Gribble, Andrew D.; Ife, Robert J.; Stevens, Nichola; Witherington, Jason Bioorganic and Medicinal Chemistry Letters, 2001 , vol. 11, # 2 p. 199 - 202

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被引用次数: 19

摘要

... Acknowledgements. The authors would like to acknowledge Thaddeus Thomaszek for determination of cathepsin K inhibition. References. 1; (a) FH Drake, RA Dodds, IE James, JR Connor, C Debouck, S Richardson, E Lee-Rykaczewski, L Coleman, D Rieman, R Barthlow, G Hastings, M Gowen; J. Biol. Chem., 271 (1996), p. 12511. ... 3; F Fenwick, B Gamier, A Gribble, R Ife, A Rawlings, J Witherington; Bioorg. Med. Chem. Lett., 11 (2000), p. 195. ...