Identification of fused bicyclic heterocycles as potent and selective 5-HT 2A receptor antagonists for the treatment of insomnia

Y Xiong, B Ullman, JSK Choi, M Cherrier…

文献索引：Bioorganic and Medicinal Chemistry Letters, , vol. 22, # 5 p. 1870 - 1873

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被引用次数: 4

摘要

... Please enable JavaScript to use all the features on this page. Bioorganic & Medicinal Chemistry Letters. ... Despite its poor metabolic stability 1 was still attractive as a chemical starting point as a result of its very favorable CNS penetration. ...