Solid-phase synthesis of indolecarboxylates using palladium-catalyzed reactions

K Yamazaki, Y Nakamura, Y Kondo

文献索引：Yamazaki, Kazuo; Nakamura, Yosuke; Kondo, Yoshinori Journal of Organic Chemistry, 2003 , vol. 68, # 15 p. 6011 - 6019

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被引用次数: 90

摘要

Polymer-supported, palladium-catalyzed cyclization reactions effectively synthesized indolecarboxylates. Palladium-catalyzed carbon-carbon bond-forming reactions of immobilized enaminoesters followed by transesterification yielded indole 2-or 3- carboxylates with various functional groups on the benzene ring. Indolecarboxylates were efficiently cyclized via an intramolecular palladium-catalyzed amination reaction of ...