Tetrahedron

Synthesis of complex fused polycyclic heterocycles utilizing IMDAF reactions of allylamino-or allyloxy-furyl (hetero) arenes

ML Read, A Krapp, PO Miranda, LL Gundersen

文献索引：Read, Matthew L.; Krapp, Andreas; Miranda, Pedro O.; Gundersen, Lise-Lotte Tetrahedron, 2012 , vol. 68, # 7 p. 1869 - 1885

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被引用次数: 19

摘要

Arenes and heteroarenes carrying a halogen and an amino-or hydroxy group have been converted to allylamino-or allyloxy-furyl-(hetero) arenes. These compounds underwent IMDAF reactions to give complex fused polycyclic heterocycles. The reactivity of the substrates was highly dependent on the detailed substitution pattern, however cyclizations occurred with high stereoselectivity in most cases. Experimental findings regarding ...