Construction of azacycles based on endo-mode cyclization of allenes

…, M Kobayashi, S Kubota, Y Takahashi…

文献索引：Mukai, Chisato; Kobayashi, Minoru; Kubota, Shoko; Takahashi, Yukie; Kitagaki, Shinji Journal of Organic Chemistry, 2004 , vol. 69, # 6 p. 2128 - 2136

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被引用次数: 29

摘要

A new procedure for constructing monocyclic five-and six-membered azacycles by the endo- mode ring-closing reaction of allenylazido derivatives under neutral conditions has been developed. The azabicyclo [mn 0] compounds were prepared by applying this newly developed procedure. The seven-membered azacycle was prepared when the allene possessing an unsubstituted carboxyl amido functionality was submitted to the basic ...