Tetrahedron letters

A synthesis of succinimides and glutarimides from cyclic anhydrides

T Kometani, T Fitz, DS Watt

文献索引：Kometani, Tadashi; Fitz, Tony; Watt, David S. Tetrahedron Letters, 1986 , vol. 27, # 8 p. 919 - 922

被引用次数: 24

摘要

Abstract The transformation of cyclic anhydrides to their corresponding imides involves a mild three-step sequence:(1) reaction with a primary amine,(2) conversion of the intermediate monoamide to an N-hydroxysuccinimidyl ester using N, N′-disuccinimidyl oxalate (DSO), and (3) cyclization by heating the NHS ester in trichloroethylene in the presence of 4-(dimethylamino) pyridine.

The Reaction of Succinic and Glutaric Acid with Amines

[Hoey; Lester Journal of the American Chemical Society, 1951 , vol. 73, p. 4473]

N-Cyanoimides: Reactivity studies with amine nucleophiles

[Stephens, Randall W.; Domeier, Linda A.; Todd, Michael G.; Nelson, Veronica A. Tetrahedron Letters, 1992 , vol. 33, # 6 p. 733 - 736]

Solvent-mediated one-pot synthesis of cyclic N-substituted i...

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N-Cyanoimides: Reactivity studies with amine nucleophiles

[Stephens, Randall W.; Domeier, Linda A.; Todd, Michael G.; Nelson, Veronica A. Tetrahedron Letters, 1992 , vol. 33, # 6 p. 733 - 736]