Discovery of orally active nonpeptide vitronectin receptor antagonists based on a 2-benzazepine Gly-Asp mimetic.
W H Miller, D P Alberts, P K Bhatnagar, W E Bondinell, J F Callahan, R R Calvo, R D Cousins, K F Erhard, D A Heerding, R M Keenan, C Kwon, P J Manley, K A Newlander, S T Ross, J M Samanen, I N Uzinskas, J W Venslavsky, C C Yuan, R C Haltiwanger, M Gowen, S M Hwang, I E James, M W Lark, D J Rieman, G B Stroup, L M Azzarano, K L Salyers, B R Smith, K W Ward, K O Johanson, W F Huffman