Organic Letters 2010-03-19

Direct and selective functionalization of a tetrahydro-beta-carboline at position 4.

Claire Rannoux, Fanny Roussi, Pascal Retailleau, Françoise Guéritte

文献索引：Org. Lett. 12(6) , 1240-3, (2010)

摘要

The first example of direct functionalization of a tetrahydro-beta-carboline (THBC) at position 4 is presented. Nucleophiles with various reactivity add to a transient intermediate generated in situ from this THBC. This reaction proceeds with a total control of the two created stereogenic centers.

结构式	名称/CAS号	分子式	全部文献
	1,2,3,4-四氢-9H-吡啶[3,4-B]并吲哚 CAS:16502-01-5	C₁₁H₁₂N₂

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Direct and selective functionalization of a tetrahydro-beta-carboline at position 4.

摘要

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