| 常用名 | 泮库溴铵 | CAS号 | 15500-66-0 |
|---|---|---|---|
| 价格 | ¥918.0/25mg ¥2818.0/100mg | 纯度 | 99.0% |
| 备货期 | 2天 | 库存 | 询单 |
| 产品详情(用途,包装等)
用途: Pancuronium Dibromide is a bis-quaternary steroid that is a competitive nicotinic antagonist.Target: nAChRPancuronium dibromide is a competitive AChR antagonist (IC50 = 5.5 nM) and acts as a skeletal muscle relaxant. Pancuronium dibromide interrupts neuromuscular transmission by competing with acetylcholine for receptor sites on the motor end-plate. Pancuronium dibromide is a non-depolarizing agent. Pancuronium is a typical non-depolarizing curare-mimetic muscle relaxant. It acts as a competitive acetylcholine antagonist on neuromuscular junctions, displacing acetylcholine (hence competitive) from its post-synaptic nicotinic acetylcholine receptors. It is (unlike suxamethonium) a non-depolarizing agent, which means that it causes no spontaneous depolarizations upon association with the nicotinic receptor in neuromuscular junction, thus producing no muscle fasciculations upon administration [1-3]. 物理化学性质: CAS号:15500-66-0 常用中文名:泮库溴铵 常用英文名:Pancuronium dibromide 分子式:C35H60Br2N2O4 分子量:732.67000 密度:N/A 沸点:N/A 熔点:214 - 217ºC 闪点:N/A 储存条件:Desiccate at RT |