Sarpogrelate hydrochloride
更新时间：2021-07-26 18:31:53
采购访问：36次
| 常用名 | 盐酸沙格雷酯 | CAS号 | 135159-51-2 |
|---|---|---|---|
| 价格 | $需询单/100g $需询单/1kg $需询单/100kg $需询单/1000kg | 纯度 | 98.0% |
| 备货期 | 需询单 | 库存 | 询单 |
| 产品详情（用途，包装等）
用途： Sarpogrelate(MCI-9042) hydrochloride, a selective 5-HT2 antagonist, has been widely used as an anti-platelet agent for the treatment of PAD.Target: 5-HT2 RecepterSarpogrelate is a drug which acts as an antagonist at the 5HT2A and 5-HT2B receptors. Sarpogrelate was shown to have the same affinity as ritanserin for 5-HT2A receptors, with a Ki value of 8.39 nM [1]. Sarpogrelate lacked prominent 5-HT1-like, 5-HT3, beta, H1, H2 and M3 antagonist activity and weakly blocked alpha 1-adrenoceptors (pKB = 6.30). (S)-M-1 showed weak affinity for 5-HT1-like receptors (pKB = 6.30), alpha 1- (pKB = 6.80) and beta- (pKB = 6.54) adrenoceptors, while (R)-M-1 was a weak antagonist at histamine H1 receptors (pKB = 6.49) [2]. After 12 weeks of sarpogrelate administration, FBF and LBF responses during RH showed significant increases from 13.2 +/- 1.7 to 18.1 +/- 2.2 mL/min per 100 mL tissue (P 物理化学性质： CAS号：135159-51-2 常用中文名：盐酸沙格雷酯 常用英文名：Sarpogrelate Hydrochloride 分子式：C24H32ClNO6 分子量：465.967 密度：N/A 沸点：585.9ºC at 760 mmHg 熔点：145-148°C 闪点：308.1ºC 储存条件：Desiccate at RT |
达阳化工（杭州）有限公司
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- 上海阿拉丁生化科技股份有限公司
- 上海市 上海市 浦东新区
- 产品名：Sarpogrelate Hydrochloride
- 价格： ￥1029.9/100mg ￥480.9/25mg ￥115.9/5mg ￥308.9/1ml
- 纯度：98.0%
- 备货期：1天
- 联系人：阿拉丁
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参考价格：$103/10mM*1mLinDMSO