依来曲普坦氢溴酸盐
更新时间：2025-09-19 00:41:51
| 常用名 | 依来曲普坦氢溴酸盐 | CAS号 | 177834-92-3 |
|---|---|---|---|
| 价格 | ￥需询单/1kg ￥需询单/1g | 纯度 | 98.0% |
| 备货期 | 3天 | 库存 | 现货 |
| 产品详情（用途，包装等）
用途： Eletriptan HBr is a selective 5-HT1B and 5-HT1D receptor agonist with Ki of 0.92 nM and 3.14 nM, respectively.IC50 value: 0.82 nM/3.14 nM (5-HT1B/5-HT1D, Ki) [1]Target: 5-HT1B/5-HT1D in vitro: [3H]Eletriptan has a total number of binding sites (Bmax) of 2478 fmol/mg and 1576 fmol/mg for 5-HT1B and 5-HT1D, respectively. [3H]Eletriptan has a significantly faster association rate (K(on) 0.249/min/nM) than [3H]sumatriptan (K(on) 0.024/min/nM) and a significantly slower off-rate (K(off) 0.027/min compared to 0.037/min for [3H]sumatriptan) [1]. Eletriptan induces concentration-dependent contractions of meningeal artery, coronary artery, and saphenous vein. The potency of Eletriptan is higher in meningeal artery than in coronary artery (86-fold) or saphenous vein (66-fold). The predicted contraction by Eletriptan (40 mg and 80 mg) and sumatriptan (100 mg) at free C(max) observed in clinical trials is similar in meningeal artery [2].in vivo: Eletriptan ( 物理化学性质： CAS号：177834-92-3 常用中文名：依来曲普坦氢溴酸盐 常用英文名：Eletriptan HBr 分子式：C22H27BrN2O2S 分子量：463.43 密度：N/A 沸点：633.9ºC at 760 mmHg 熔点：169-171ºC 闪点：337.2ºC 储存条件：Desiccate at RT |
- 上海阿拉丁生化科技股份有限公司
- 上海市 上海市 浦东新区
- 产品名：Eletriptan HBr
- 价格： ￥92.9/10mg ￥339.9/250mg ￥175.9/50mg ￥504.9/1g
- 纯度：98.0%
- 备货期：1天
- 联系人：阿拉丁
- 上海阿摩尔生物科技有限公司
- 上海市 上海市 奉贤区
- 产品名：(R)-3-((1-甲基-2-吡咯烷基)甲基)-5-(2-(苯磺酰)乙基)-1H-吲哚氢溴酸盐
- 价格： ￥需询单/100mg ￥需询单/1g ￥需询单/250mg ￥需询单/50mg
- 纯度：98.0%
- 备货期：需询单
- 联系人：王汐瑶
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参考价格：$84/5mg