| 常用名 | BET bromodomain inhibitor 1 | CAS号 | 2411226-02-1 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: BET bromodomain inhibitor 1 is an orally active, selective bromodomain and extra-terminal (BET) bromodomain inhibitor with an IC50 of 2.6 nM for BRD4. BET bromodomain inhibitor 1 binds to BRD2(2), BRD3(2), BRD4(1), BRD4(2), and BRDT(2) with high affinities (Kd values of 1.3 nM, 1.0 nM, 3.0 nM, 1.6 nM, 2.1 nM, respectively). bromodomain inhibitor 1 has anti-cancer activity[1]. 物理化学性质: CAS号:2411226-02-1 常用中文名:BET bromodomain inhibitor 1 常用英文名:BET bromodomain inhibitor 1 分子式:C22H19F2N3O4S 分子量:459.47 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A |