| 常用名 | BI-2865 | CAS号 | 2937327-93-8 |
|---|---|---|---|
| 价格 | 纯度 | 99.39% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: BI-2865 is a none-covalent pan-KRAS Inhibitor. BI-2865 binds to WT, G12C, G12D, G12V and G13D mutant KRAS with KDs of 6.9, 4.5, 32, 26, 4.3 nM respectively. BI-2865 inhibits the proliferation of G12C, G12D or G12V mutant KRAS expressing BaF3 cells (mean IC50: roughly 140 nM)[1]. 物理化学性质: CAS号:2937327-93-8 常用中文名:BI-2865 常用英文名:BI-2865 分子式:C23H27N7O2S 分子量:465.57 密度:1.38±0.1 g/cm3(Temp: 20 °C; Press: 760 Torr)(Predicted) 沸点:708.7±70.0 °C(Predicted) 熔点:N/A 闪点:N/A |