| 常用名 | NVP-MELK8a hydrochloride | CAS号 | 2096992-20-8 |
|---|---|---|---|
| 价格 | 纯度 | 98.0% | |
| 备货期 | 10天 | 库存 | 现货 |
| 产品详情(用途,包装等)
用途: NVP-MELK8a hydrochloride (MELK8a hydrochloride) is a novel potent, and selective MELK inhibitor with IC50 of 2 nM; exhibits high selectivity with only 7 off-target kinases inhibited >85% against 456 kinases at 1 uM, Flt3 (IC50=0.18 uM), Haspin (IC50=0.19 uM), PDGFRα (IC50=0.42 uM); exhibits growth inhibition of MDA-MD-468 cells with IC50 of 0.11 uM, and increases cells harboring 4N DNA content. 物理化学性质: CAS号:2096992-20-8 常用中文名:NVP-MELK8a hydrochloride 常用英文名:NVP-MELK8a hydrochloride 分子式:C25H33ClN6O 分子量:469.02212 密度:N/A 沸点:N/A 熔点:N/A 闪点:N/A 储存条件:2-8℃ |