129888-60-4

• 常用中文名：N-BOC-3-甲磺酰氧基哌啶
• 常用英文名：N-Boc-3-mesyloxypiperidine
• CAS号：129888-60-4
• 分子式：C₁₁H₂₁NO₅S
• 分子量：279.353
• 发布时间：2018-06-17 12:51:39
• 更新时间：2026-07-06 18:38:56

名称

• 中文名: N-BOC-3-甲磺酰氧基哌啶
• 英文名: N-Boc-3-mesyloxypiperidine
• 中文别名: N-BOC-3-甲磺酰氧基哌啶N-BOC-3-甲磺酰氧基哌啶; 3-((甲磺酰基)氧基)哌啶-1-甲酸叔丁酯; 3-(甲基磺酰基氧基)哌啶-1-羧酸叔丁酯; 1-BOC-3-[(甲磺酰基)氧基]哌啶; N-BOC-3-OMS-哌啶; N-Boc-3-甲基磺酰氧基哌啶
• 英文别名: tert-Butyl 3-[(methylsulfonyloxy)]-1-piperidinecboxylate; tert-Butyl 3-((methylsulfonyl); 2-Methyl-2-propanyl 3-[(methylsulfonyl)oxy]-1-piperidinecarboxylate; tert-Butyl 3-Methylsulfonyloxypiperidine-1-carboxylate; tert-Butyl 3-(methanesulfonyloxy)piperidine-1-cboxylate; 1-Boc-3-methanesulphonyloxypiperidine; tert-Butyl 3-Methylsulfonyloxypiperidine-1-cboxylate; 3-((methylsulfonyl)oxy)piperidine-1-cboxylate; tert-Butyl 3-[(methylsulfonyl)oxy]piperidine-1-carboxylate; tert-Butyl 3-Methylsulfonyloxypiperidin-1-carboxylate; N-BOC-3-(Methylsulfonyloxy)piperidine; 1,1-Dimethylethyl 3-[(methylsulfonyl)oxy]-1-piperidinecboxylate; 3-(Methylsulfonyloxy)piperidine-1-cboxylic acid tert-butyl ester; tert-Butyl 3-((methylsulfonyl)oxy)piperidine-1-carboxylate; 1-Boc-3-methanesulfonyloxy-piper; 1-Piperidinecboxylic acid, 3-[(Methylsulfonyl)oxy]-, 1,1-diMethylethyl ester; 3-methylsulfonyloxy-1-piperidinecboxylic acid tert-butyl ester; 3-methanesulfonyloxy-N-t-butoxycarbonylpiperidine; 1-Piperidinecarboxylic acid, 3-[(methylsulfonyl)oxy]-, 1,1-dimethylethyl ester; tert-Butyl 3-Methylsulfonyloxypiperidin-1-cboxylate; tert-Butyl 3-[(methylsulfonyl)oxy]-1-piperidinecarboxylate; 1-(tert-Butoxycbonyl)-3-(methanesulfonyloxy)piperidine; 1-tert-butoxycarbonylpiperid-3-yl methanesulfonate

物化性质

• 密度: 1.2±0.1 g/cm3
• 沸点: 407.2±34.0 °C at 760 mmHg
• 分子式: C₁₁H₂₁NO₅S
• 分子量: 279.353
• 闪点: 200.1±25.7 °C
• 精确质量: 279.114044
• PSA: 81.29000
• LogP: 0.64
• 蒸汽压: 0.0±0.9 mmHg at 25°C
• 折射率: 1.500
• 储存条件: 室温，干燥

安全

• 海关编码: 2933399090

合成路线

85275-45-2 124-63-0 ~99% 129888-60-4

文献：VERTEX PHARMACEUTICALS INCORPORATED; Charrier, Jean-Damien; Durrant, Steven John; Knegtel, Ronald Patent: US2013/115310 A1, 2013 ; Location in patent: Paragraph 0248; 0249 ;

85275-45-2 7143-01-3 ~90% 129888-60-4

文献：BIOGEN IDEC MA INC.; SUNESIS PHARMACEUTICALS, INC.; HOPKINS, Brian, T.; SCOTT, Daniel; CONLON, Patrick; JENKINS, Tracy, J.; POWELL, Noel; GUAN, Bing; CURERVO, Julio, H.; WANG, Deping; TAVERAS, Art Patent: WO2012/58645 A1, 2012 ; Location in patent: Page/Page column 210 ; WO 2012/058645 A1

85275-45-2 124-63-0 121-44-8 ~94% 129888-60-4

文献：The United States of America as represented by the Department of Health and Human Services Patent: US5571832 A1, 1996 ; US 5571832 A

6859-99-0 ~% 129888-60-4

文献：Journal of Medicinal Chemistry, , vol. 35, # 23 p. 4334 - 4343

24424-99-5 ~% 129888-60-4

文献：Journal of Medicinal Chemistry, , vol. 35, # 23 p. 4334 - 4343

上下游产品

上游产品  6
85275-45-2 124-63-0 7143-01-3 121-44-8
6859-99-0 24424-99-5
下游产品  5
131667-57-7 85838-94-4 5810-55-9 129888-61-5
144243-24-3

海关

海关编码	2933399090
中文概述	2933399090. 其他结构含非稠合吡啶环的化合物. 增值税率:17.0%. 退税率:13.0%. 监管条件:无. 最惠国关税:6.5%. 普通关税:20.0%
申报要素	品名, 成分含量, 用途, 乌洛托品请注明外观, 6－己内酰胺请注明外观, 签约日期
Summary	2933399090. other compounds containing an unfused pyridine ring (whether or not hydrogenated) in the structure. VAT:17.0%. Tax rebate rate:13.0%. . MFN tariff:6.5%. General tariff:20.0%