202477-59-6

• 常用中文名：(2S,4R)-1-(叔丁氧羰基)-4((甲磺酰基)氧基)吡咯烷-2-羧酸
• 常用英文名：(2S,4R)-1-(TERT-BUTOXYCARBONYL)-4-((METHYLSULFONYL)OXY)PYRROLIDINE-2-CARBOXYLIC ACID
• CAS号：202477-59-6
• 分子式：C₁₁H₁₉NO₇S
• 分子量：309.33600
• 发布时间：2018-12-10 08:46:46
• 更新时间：2026-07-28 19:50:42

名称

• 中文名: (2S,4r)-1-boc-4-甲磺酰氧基脯氨酸
• 英文名: (2S,4R)-1-[(2-methylpropan-2-yl)oxycarbonyl]-4-methylsulfonyloxypyrrolidine-2-carboxylic acid
• 中文别名: N-BOC-反式-4-甲磺酰基-L-脯氨酸; (2S,4R)-4-[(甲磺酰基)氧基]-1,2-吡咯烷二甲酸 1-叔丁酯/202-6; (2S,4R)-4-[(甲磺酰基)氧基]-1,2-吡咯烷二甲酸 1-叔丁酯; (2S,4R)-1-BOC-4-甲磺酰氧基脯氨酸
• 英文别名: (2S,4R)-1-BOC-4-METHANESULFONYLOXY-PROLINE; (2S,4R)-1-[(2-methylpropan-2-yl)oxycbonyl]-4-methylsulfonyloxypyrrolidine-2-cboxylic acid; (2S,4R)-1-t-butoxycbonyl-4-methanesulfon yloxypyrrolidine-2-cboxylic acid; (2S,4R)-1-(tert-Butoxycbonyl)-4-((methylsulfonyl)oxy)pyrrolidine-2-cboxylic acid; (2S,4R)-4-Methanesulfonyloxy-pyrrolidine-1,2-dicboxylic acid 1-tert-butyl ester; (2S,4R)-4-Methanesulfonyloxy-pyrrolidine-1,2-dicarboxylic acid 1-tert-butyl ester; (2S,4R)-1-(tert-Butoxycarbonyl)-4-((methylsulfonyl)oxy)pyrrolidine-2-carboxylic acid; (2S,4R)-1-(tert-butoxycarbonyl)-4-[(methylsulfonyl)oxy]-2-pyrrolidinecarboxylic acid; (2S,4R)-1-Boc-4-methanesulfonyloxy-proline; 1,2-Pyrrolidinedicboxylic acid, 4-[(methylsulfonyl)oxy]-, 1-(1,1-dimethylethyl) ester, (2S,4R); N-Boc-(2S,4R)-4-mesylproline; (2S,4R)-4-[(Methylsulfonyl)oxy]-1,2-pyrrolidinedicboxylic acid 1-(1,1-dimethylethyl) ester; (2S,4R)-N-Boc-trans-4-methanesulfonyloxy-L-proline

物化性质

• 密度: 1.38g/cm3
• 沸点: 500.1ºC at 760 mmHg
• 分子式: C₁₁H₁₉NO₇S
• 分子量: 309.33600
• 闪点: 256.3ºC
• 精确质量: 309.08800
• PSA: 118.59000
• LogP: 1.44390
• 蒸汽压: 2.32E-11mmHg at 25°C
• 折射率: 1.528
• 储存条件: 2-8°C

合成路线

84520-67-2 ~87% 202477-59-6

文献：Lange, Udo E.W.; Baucke, Dorit; Hornberger, Wilfried; Mack, Helmut; Seitz, Werner; Hoeffken, H. Wolfgang Bioorganic and Medicinal Chemistry Letters, 2006 , vol. 16, # 10 p. 2648 - 2653

13726-69-7 124-63-0 ~% 202477-59-6

文献：Chorghade, Mukund S.; Mohapatra, Debendra K.; Sahoo, Gokarneswar; Gurjar, Mukund K.; Mandlecha, Manish V.; Bhoite, Nitin; Moghe, Santosh; Raines, Ronald T. Journal of Fluorine Chemistry, 2008 , vol. 129, # 9 p. 781 - 784

13726-69-7 ~% 202477-59-6

文献：Bernard, Harald; Buelow, Gerd; Lange, Udo E. W.; Mack, Helmut; Pfeiffer, Thomas; Schaefer, Bernd; Seitz, Werner; Zierke, Thomas Synthesis, 2004 , # 14 p. 2367 - 2375

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