191092-07-6

• 常用中文名：(R)-3-(甲苯磺酰氧基甲基)哌啶-1-羧酸叔丁酯
• 常用英文名：(R)-3-(Tosyloxymethyl)-N-Boc-piperidine
• CAS号：191092-07-6
• 分子式：C₁₈H₂₇NO₅S
• 分子量：369.47600
• 发布时间：2018-10-08 13:22:20
• 更新时间：2024-01-11 07:47:15

名称

• 中文名: (R)-3-(甲苯磺酰氧基甲基)哌啶-1-羧酸叔丁酯
• 英文名: (R)-3-(Tosyloxymethyl)-N-Boc-piperidine
• 英文别名: tert-butyl (3R)-3-({[(4-methylphenyl)sulfonyl]oxy}methyl)piperidine-1-carboxylate; 3-(BOC-AMINO)PYRROLIDINE HYDROCHLORIDE; 3-(tert-butoxycarbonyl-amino)pyrrolidine; 3-(N-tert-butoxycarbonylamino)pyrrolidine; 1,1-dimethylethyl (3R)-3-({[(4-methylphenyl)sulfonyl]oxy}methyl)-1-piperidinecarboxylate; tert-butyl 3-pyrrolidinylcarbamate; (R)-tert-butyl 3-((tosyloxy)methyl)piperidine-1-carboxylate; tert-butyl (R)-3-(tosyloxymethyl)piperidine-1-carboxylate; pyrrolidin-3-ylcarbamic acid tert-butyl ester; 3-(BOC-amino)pyrrolidine; 1,1-dimethylethyl (3-pyrrolidinyl)carbamate; BOC-(+/-)-(3)APYROLIDI; 3-N-BOC-AMINO PYRROLIDINE; 3-N-Boc-aMinoMethypyrrolidine; BOC-(+/-)-3-AMINOPYRROLIDINE; 3-Aminopyrrolidine,3-BOC protected

物化性质

• 分子式: C₁₈H₂₇NO₅S
• 分子量: 369.47600
• 精确质量: 369.16100
• PSA: 81.29000
• LogP: 4.36610

合成路线

116574-71-1 98-59-9 ~92% 191092-07-6

文献：SMITHKLINE BEECHAM CORPORATION Patent: WO2008/157330 A1, 2008 ; Location in patent: Page/Page column 92 ;

25137-01-3 ~% 191092-07-6

文献：Rivera, Jocelyn; Jayasuriya, Nilukshi; Rane, Dinanath; Keertikar; Ferreira, J.Albert; Chao, Jianping; Minor, Keith; Guzi, Timothy Tetrahedron Letters, 2002 , vol. 43, # 49 p. 8917 - 8919

4124-41-8 116574-71-1 ~% 191092-07-6

文献：Prabhakaran, Jaya; Arango, Victoria; Majo, Vattoly J.; Simpson, Norman R.; Kassir, Suham A.; Underwood, Mark D.; Polavarapu, Hanish; Bruce, Jeffrey N.; Canoll, Peter; John Mann; Dileep Kumar Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 15 p. 5104 - 5107

37675-20-0 ~% 191092-07-6

文献：Rivera, Jocelyn; Jayasuriya, Nilukshi; Rane, Dinanath; Keertikar; Ferreira, J.Albert; Chao, Jianping; Minor, Keith; Guzi, Timothy Tetrahedron Letters, 2002 , vol. 43, # 49 p. 8917 - 8919