马扎哌汀

• 常用名: 马扎哌汀
• 英文名: Mazapertine
• CAS号: 134208-17-6
• 分子量: 421.57500
• 密度: 1.128g/cm3
• 沸点: 583.8ºC at 760 mmHg
• 分子式: C₂₆H₃₅N₃O₂
• 熔点: N/A
• 闪点: 306.9ºC

马扎哌汀名称

• 中文名: 马扎哌汀
• 英文名: piperidin-1-yl-[3-[[4-(2-propan-2-yloxyphenyl)piperazin-1-yl]methyl]phenyl]methanone

马扎哌汀物理化学性质

• 密度: 1.128g/cm3
• 沸点: 583.8ºC at 760 mmHg
• 分子式: C₂₆H₃₅N₃O₂
• 分子量: 421.57500
• 闪点: 306.9ºC
• 精确质量: 421.27300
• PSA: 36.02000
• LogP: 4.36290
• InChIKey: ZKZFPRUSWCYSGT-UHFFFAOYSA-N
• SMILES: CC(C)Oc1ccccc1N1CCN(Cc2cccc(C(=O)N3CCCCC3)c2)CC1
• 蒸汽压: 1.29E-13mmHg at 25°C
• 折射率: 1.584

马扎哌汀靶点实验

查看更多实验

实验名称：The compound is evaluated for inhibition of apomorphine induced climbing behavior in ... 来源：ChEMBL 靶标：Mus musculus External Id：CHEMBL716324

实验名称：The compound is evaluated for inhibition of apomorphine induced emesis in dogs after ... 来源：ChEMBL 靶标：Canis lupus familiaris External Id：CHEMBL667134

实验名称：Binding affinity towards 5-hydroxytryptamine 1A receptor of rat brain synaptosomal pr... 来源：ChEMBL 靶标：5-hydroxytryptamine receptor 1A External Id：CHEMBL616580

实验名称：Volume of distribution at steady state in human at 2.8 mg, iv 来源：ChEMBL 靶标：Homo sapiens External Id：CHEMBL1028548

实验名称：The compound is evaluated for inhibition of apomorphine induced emesis in dogs after ... 来源：ChEMBL 靶标：Canis lupus familiaris External Id：CHEMBL667135

实验名称：The compound is evaluated for inhibition of 8-OH-DPAT induced reciprocal forepaw trea... 来源：ChEMBL 靶标：Rattus norvegicus External Id：CHEMBL784411

实验名称：Binding affinity towards alpha-1 adrenergic receptor using [3H]prazosin as radioligan... 来源：ChEMBL 靶标：Alpha-1A adrenergic receptor External Id：CHEMBL649341

实验名称：Binding affinity was determined against 5-hydroxytryptamine 1A receptor using [3H]WB-... 来源：ChEMBL 靶标：5-hydroxytryptamine receptor 1A External Id：CHEMBL616088

实验名称：Compound was measured in vivo for its binding affinity at Alpha-1 adrenergic receptor... 来源：ChEMBL 靶标：Alpha-1B adrenergic receptor External Id：CHEMBL648824

实验名称：Compound was measured for its antipsychotic activity in the rat conditioned avoidance... 来源：ChEMBL 靶标：Rattus norvegicus External Id：CHEMBL785347

共43条，当前第1页，共5页

1

2

3

4

5

马扎哌汀英文别名

• UNII-N0X1XW704P
• [3-[[4-[2-(1-Methylethoxy)phenyl]-1-piperazinyl]methyl]benzoyl]-piperidine
• Mazapertine
• Mazapertine [INN]
• 1-[3-[[4-[2-(1-methylethoxy)phenyl]-1-piperazinyl]methyl]benzoyl]piperidine