Lassbio-1359

• 常用名: Lassbio-1359
• 英文名: Lassbio-1359
• CAS号: 1396397-19-5
• 分子量: 298.34
• 密度: N/A
• 沸点: N/A
• 分子式: C₁₇H₁₈N₂O₃
• 熔点: N/A
• 闪点: N/A

Lassbio-1359用途

LASSBio-1359是一种腺苷受体激动剂。它的作用是诱导海绵体松弛。它也是一种新型的选择性磷酸二酯酶。

Lassbio-1359名称

• 英文名: LASSBio-1359

Lassbio-1359生物活性

• 描述: LASSBio-1359是一种腺苷受体激动剂。它的作用是诱导海绵体松弛。它也是一种新型的选择性磷酸二酯酶。
• 参考文献: 1. Montes GC, Hammes N, da Rocha MD, Montagnoli TL, Fraga CA, Barreiro EJ, Sudo RT, Zapata-Sudo G. Treatment with Adenosine Receptor Agonist Ameliorates Pain Induced by Acute and Chronic Inflammation. J Pharmacol Exp Ther. 2016 Aug;358(2):315-23. doi: 10.1124/jpet.115.231241. Epub 2016 May 18. PubMed PMID: 27194479.

Lassbio-1359物理化学性质

• 分子式: C₁₇H₁₈N₂O₃
• 分子量: 298.34
• InChIKey: ZKKIMIBBUMDNHP-LDADJPATSA-N
• SMILES: COc1ccc(C=NN(C)C(=O)c2ccccc2)cc1OC

Lassbio-1359靶点实验

查看更多实验

实验名称：Inhibition of bovine PDE4 using [3H]cAMP as substrate at 10 uM 来源：ChEMBL 靶标：N/A External Id：CHEMBL2175864

实验名称：Antiinflammatory activity in A/J mouse assessed as inhibition of LPS-induced airway r... 来源：ChEMBL 靶标：Mus musculus External Id：CHEMBL2175723

实验名称：Inhibition of bovine PDE4 using [3H]cAMP as substrate 来源：ChEMBL 靶标：N/A External Id：CHEMBL2175863

实验名称：Antiinflammatory activity in A/J mouse assessed as inhibition of leukocyte accumulati... 来源：ChEMBL 靶标：Mus musculus External Id：CHEMBL2175730

实验名称：Antiinflammatory activity in A/J mouse assessed as inhibition of neutrophil accumulat... 来源：ChEMBL 靶标：Mus musculus External Id：CHEMBL2175728

实验名称：Inhibition of bovine PDE1 using [3H]cAMP as substrate at 10 uM 来源：ChEMBL 靶标：N/A External Id：CHEMBL2175749

实验名称：Inhibition of human PDE2 using [3H]cAMP as substrate at 10 uM 来源：ChEMBL 靶标：cGMP-dependent 3',5'-cyclic phosphodiesterase External Id：CHEMBL2175747

实验名称：Antiinflammatory activity in A/J mouse assessed as inhibition of LPS-induced airway e... 来源：ChEMBL 靶标：Mus musculus External Id：CHEMBL2175604

实验名称：Inhibition of PDE6 at 10 uM 来源：ChEMBL 靶标：N/A External Id：CHEMBL2175742

实验名称：Selectivity ratio of IC50 for bovine PDE3 to IC50 for bovine PDE4 来源：ChEMBL 靶标：N/A External Id：CHEMBL2175739

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