PF-06649298

更新时间：2026-05-12 12:05:30

PF-06649298结构式	常用名	PF-06649298	英文名	PF-06649298
	CAS号	1854061-16-7	分子量	294.347
	密度	N/A	沸点	N/A
	分子式	C₁₆H₂₂O₅	熔点	N/A
	MSDS	N/A	闪点	N/A

PF-06649298用途

PF-06649298(PF06649298)Na+/柠檬酸转运蛋白NaCT(SLC13A5)的有效选择性抑制剂,显示抑制HEKNaCT细胞中柠檬酸盐的摄取,IC50为0.41 uM；显示出比NaDC1和NaDC3高>60倍的选择性。

英文名	PF-06649298

描述	PF-06649298(PF06649298)Na+/柠檬酸转运蛋白NaCT(SLC13A5)的有效选择性抑制剂,显示抑制HEKNaCT细胞中柠檬酸盐的摄取,IC50为0.41 uM；显示出比NaDC1和NaDC3高>60倍的选择性。
参考文献	References 1. Pajor AM, et al. Mol Pharmacol. 2016 Dec;90(6):755-765. View Related Products by Target Sodium-coupled Citrate Transporter (NaCT,SLC13A5)

分子式	C₁₆H₂₂O₅
分子量	294.347

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