3,4-Piperidinediol, 5-(hydroxymethyl)-, (3R,4R,5S)- (9CI)

• 常用名: 3,4-Piperidinediol, 5-(hydroxymethyl)-, (3R,4R,5S)- (9CI)
• 英文名: 3,4-Piperidinediol, 5-(hydroxymethyl)-, (3R,4R,5S)- (9CI)
• CAS号: 202979-51-9
• 分子量: 147.17200
• 密度: N/A
• 沸点: N/A
• 分子式: C₆H₁₃NO₃
• 熔点: N/A
• 闪点: N/A

用途

L-Afegostat(5-epi-Isofagomine)是一种糖苷酶抑制剂。L-Afegostat是一种亚氨基糖,可用于合成碳水化合物。L-Afegostat显示出对β-葡萄糖苷酶的酶抑制作用,Ki为30μM[1]。

名称

• 英文名: (3R,4R,5S)-5-(hydroxymethyl)piperidine-3,4-diol

生物活性

• 描述: L-Afegostat(5-epi-Isofagomine)是一种糖苷酶抑制剂。L-Afegostat是一种亚氨基糖,可用于合成碳水化合物。L-Afegostat显示出对β-葡萄糖苷酶的酶抑制作用,Ki为30μM[1]。
• 相关类别:
  研究领域 >> 代谢疾病
• 参考文献:

  [1]. Pandey G, et al. A new access to polyhydroxy piperidines of the azasugar class: synthesis and glycosidase inhibition studies. Org Biomol Chem. 2003 Oct 7;1(19):3321-6.

物理化学性质

• 分子式: C₆H₁₃NO₃
• 分子量: 147.17200
• 精确质量: 147.09000
• PSA: 72.72000
• InChIKey: QPYJXFZUIJOGNX-KVQBGUIXSA-N
• SMILES: OCC1CNCC(O)C1O

靶点实验

查看更多实验

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英文别名

• 5-epi-Isofagomine