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ASGPR modulator-1

更新时间:2025-10-09 13:15:37

ASGPR modulator-1结构式
ASGPR modulator-1结构式
品牌特惠专场
常用名 ASGPR modulator-1 英文名 ASGPR modulator-1
CAS号 2052968-88-2 分子量 527.62
密度 N/A 沸点 N/A
分子式 C29H33N7O3 熔点 N/A
MSDS N/A 闪点 N/A

 ASGPR modulator-1用途


ASGPR调节剂-1(化合物5TJX)是一种大环化合物,可用于蛋白质-蛋白质相互作用研究[1]。

 ASGPR modulator-1名称

英文名 ASGPR modulator-1

 ASGPR modulator-1生物活性

描述 ASGPR调节剂-1(化合物5TJX)是一种大环化合物,可用于蛋白质-蛋白质相互作用研究[1]。
相关类别
参考文献

[1]. Sarah J Martin, et al. Modelling the binding mode of macrocycles: Docking and conformational sampling. Bioorg Med Chem. 2020 Jan 1;28(1):115143.

 ASGPR modulator-1物理化学性质

分子式 C29H33N7O3
分子量 527.62

 ASGPR modulator-1靶点实验

查看更多实验

实验名称:Apparent permeability across MDCK cells at 1 uM
来源:ChEMBL
靶标:NON-PROTEIN TARGET
External Id:CHEMBL3877115
实验名称:Half life in rat liver microsomes in presence of NADPH by LC/MS/MS analysis
来源:ChEMBL
靶标:N/A
External Id:CHEMBL3877131
实验名称:Selectivity ratio of IC50 for bovine trypsin to IC50 for human plasma kallikrein
来源:ChEMBL
靶标:N/A
External Id:CHEMBL3877121
实验名称:Inhibition of human plasma kallikrein using D-Pro-Phe-Arg-pNA as substrate preincubat...
来源:ChEMBL
靶标:Plasma kallikrein
External Id:CHEMBL3877122
实验名称:Inhibition of human plasma kallikrein incubated for 1 hrs
来源:ChEMBL
靶标:Plasma kallikrein
External Id:CHEMBL5234019
实验名称:Selectivity ratio of IC50 for factor 12a (unknown origin) to IC50 for human plasma ka...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL3877117
实验名称:Selectivity ratio of IC50 for tPA (unknown origin) to IC50 for human plasma kallikrei...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL3877118
实验名称:Selectivity ratio of IC50 for factor 10a (unknown origin) to IC50 for human plasma ka...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL3877119
实验名称:Selectivity ratio of IC50 for plasmin (unknown origin) to IC50 for human plasma kalli...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL3877120
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