(R)-N-(4-(4-(3-Chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl)-3-hydroxybutyl)-1H-indole-2-carboxamide

• 常用名: (R)-N-(4-(4-(3-Chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl)-3-hydroxybutyl)-1H-indole-2-carboxamide
• 英文名: (R)-N-(4-(4-(3-Chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl)-3-hydroxybutyl)-1H-indole-2-carboxamide
• CAS号: 2133454-49-4
• 分子量: 485.0
• 密度: N/A
• 沸点: N/A
• 分子式: C₂₆H₃₃ClN₄O₃
• 熔点: N/A
• 闪点: N/A

名称

• 英文名: (R)-N-(4-(4-(3-Chloro-5-ethyl-2-methoxyphenyl)piperazin-1-yl)-3-hydroxybutyl)-1H-indole-2-carboxamide

物理化学性质

• 分子式: C₂₆H₃₃ClN₄O₃
• 分子量: 485.0
• InChIKey: NRSBRNRWCATXOT-HXUWFJFHSA-N
• SMILES: CCC1=CC(=C(C(=C1)Cl)OC)N2CCN(CC2)C[C@@H](CCNC(=O)C3=CC4=CC=CC=C4N3)O

靶点实验

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实验名称：Selectivity ratio of Ki for displacement of [3H]N-methylspiperone from human D2L rece... 来源：ChEMBL 靶标：N/A External Id：CHEMBL4415926

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实验名称：Radioligand Binding Assay from US Patent US11337971: "Dopamine D3 receptor selective ... 来源：BindingDB 靶标：N/A External Id：BindingDB_10614_1

实验名称：Tmax in Long-Evans rat brain at 10 mg/kg, po measured up to 24 hrs by LC/MS/MS analys... 来源：ChEMBL 靶标：N/A External Id：CHEMBL4415942

实验名称：AUC (0 to t) in Long-Evans rat plasma at 10 mg/kg, po measured up to 24 hrs by LC/MS/... 来源：ChEMBL 靶标：N/A External Id：CHEMBL4415943

实验名称：AUC (0 to t) in Long-Evans rat brain at 10 mg/kg, po measured up to 24 hrs by LC/MS/M... 来源：ChEMBL 靶标：N/A External Id：CHEMBL4415944

实验名称：Ratio of AUC (0 to t) in Long-Evans rat brain to plasma at 10 mg/kg, po measured up t... 来源：ChEMBL 靶标：N/A External Id：CHEMBL4415945

实验名称：Ratio of drug level in Long-Evans rat brain at 10 mg/kg, po measured 8 hrs post dose ... 来源：ChEMBL 靶标：N/A External Id：CHEMBL4415946

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实验名称：Selectivity ratio of Ki for displacement of [125I] DOI from 5HT2A receptor (unknown o... 来源：ChEMBL 靶标：N/A External Id：CHEMBL4415936

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