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PF-06882961

更新时间:2025-08-25 18:14:14

PF-06882961结构式
PF-06882961结构式
品牌特惠专场
常用名 PF-06882961 英文名 PF-06882961
CAS号 2230198-02-2 分子量 555.60
密度 N/A 沸点 N/A
分子式 C31H30FN5O?4 熔点 N/A
MSDS N/A 闪点 N/A

 PF-06882961用途


PF-06882961是胰高血糖素样肽-1受体(GLP-1R)的有效的口服生物可利用激动剂。

 PF-06882961名称

英文名 PF-06882961

 PF-06882961生物活性

描述 PF-06882961是胰高血糖素样肽-1受体(GLP-1R)的有效的口服生物可利用激动剂。

 PF-06882961物理化学性质

分子式 C31H30FN5O?4
分子量 555.60
储存条件 -20°C,密闭,干燥

 PF-06882961靶点实验

查看更多实验

实验名称:In vivo agonist activity at GLP-1R in C57BL/6J mouse with human GLP-1R knock-in asses...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL5344110
实验名称:Partial agonist activity at N-terminal HA-tagged human GLP-1R expressed in HEK293 cel...
来源:ChEMBL
靶标:Glucagon-like peptide 1 receptor
External Id:CHEMBL5344107
实验名称:In vivo agonist activity at GLP-1R in C57BL/6J mouse with human GLP-1R knock-in asses...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL5344108
实验名称:Partial agonist activity at N-terminal HA-tagged human GLP-1R expressed in HEK293 cel...
来源:ChEMBL
靶标:Glucagon-like peptide 1 receptor
External Id:CHEMBL5344105
实验名称:Agonist activity at N-terminal HA-tagged human GLP-1R expressed in HEK293 cells asses...
来源:ChEMBL
靶标:Glucagon-like peptide 1 receptor
External Id:CHEMBL5344103
实验名称:Agonist activity at N-terminal HA-tagged human GLP-1R expressed in HEK293 cells asses...
来源:ChEMBL
靶标:Glucagon-like peptide 1 receptor
External Id:CHEMBL5344101
实验名称:Activation of mouse GLP-1R
来源:ChEMBL
靶标:Glucagon-like peptide 1 receptor
External Id:CHEMBL5344096
实验名称:Agonist activity human GLP-1R stably expressed in HEK293 cells assessed as reduction ...
来源:ChEMBL
靶标:Glucagon-like peptide 1 receptor
External Id:CHEMBL5552312
实验名称:Stability in rat liver microsomes assessed as intrinsic clearance at 1 uM measured up...
来源:ChEMBL
靶标:N/A
External Id:CHEMBL5344091
实验名称:Agonist activity human GLP-1R stably expressed in HEK293 cells assessed as reduction ...
来源:ChEMBL
靶标:Glucagon-like peptide 1 receptor
External Id:CHEMBL5552313
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