KB-0742 盐酸盐

• 常用名: KB-0742 盐酸盐
• 英文名: KB-0742 HCl
• CAS号: 2416873-83-9
• 分子量: 287.4
• 密度: N/A
• 沸点: N/A
• 分子式: C₁₆H₂₅N₅
• 熔点: N/A
• 闪点: N/A

KB-0742 盐酸盐用途

KB-0742是一种口服生物利用的选择性CDK9抑制剂,在CRPC模型中具有强大的抗肿瘤活性。

KB-0742 盐酸盐名称

• 中文名: KB-0742 盐酸盐
• 英文名: KB-0742 HCl

KB-0742 盐酸盐生物活性

• 描述: KB-0742是一种口服生物利用的选择性CDK9抑制剂,在CRPC模型中具有强大的抗肿瘤活性。

KB-0742 盐酸盐物理化学性质

• 分子式: C₁₆H₂₅N₅
• 分子量: 287.4
• InChIKey: VYKCLMALANGCDF-STQMWFEESA-N
• SMILES: CCC(CC)c1cc(NC2CCC(N)C2)n2nccc2n1
• 储存条件: 2-8℃

KB-0742 盐酸盐靶点实验

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实验名称：Selectivity index, ratio of IC50 for inhibition of human CDK4/Cyclin D1 to IC50 for i... 来源：ChEMBL 靶标：N/A External Id：CHEMBL5376184

实验名称：Selectivity index, ratio of IC50 for inhibition of human CDK7/Cyclin H to IC50 for in... 来源：ChEMBL 靶标：N/A External Id：CHEMBL5376185

实验名称：Inhibition of human CDK7/Cyclin H preincubated for 20 mins followed by 32P-ATP additi... 来源：ChEMBL 靶标：Cyclin-H External Id：CHEMBL5376182

实验名称：Inhibition of human CDK8/Cyclin C preincubated for 20 mins followed by 32P-ATP additi... 来源：ChEMBL 靶标：Cyclin-C External Id：CHEMBL5376183

实验名称：Inhibition of human CDK5/P25 preincubated for 20 mins followed by 32P-ATP addition an... 来源：ChEMBL 靶标：Cyclin-dependent kinase 5 External Id：CHEMBL5376180

实验名称：Inhibition of human CDK6/Cyclin D1 preincubated for 20 mins followed by 32P-ATP addit... 来源：ChEMBL 靶标：Cyclin-dependent kinase 6 External Id：CHEMBL5376181

实验名称：Inhibition of human CDK3/Cyclin E preincubated for 20 mins followed by 32P-ATP additi... 来源：ChEMBL 靶标：G1/S-specific cyclin-E1 External Id：CHEMBL5376178

实验名称：Inhibition of human CDK4/Cyclin D1 preincubated for 20 mins followed by 32P-ATP addit... 来源：ChEMBL 靶标：Cyclin-dependent kinase 4 External Id：CHEMBL5376179

实验名称：Inhibition of human CDK1/Cyclin A preincubated for 20 mins followed by 32P-ATP additi... 来源：ChEMBL 靶标：Cyclin-dependent kinase 1 External Id：CHEMBL5376176

实验名称：Inhibition of human CDK2/Cyclin A preincubated for 20 mins followed by 32P-ATP additi... 来源：ChEMBL 靶标：Cyclin-A1 External Id：CHEMBL5376177

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