cyclopropyl[4-(2-{2-[(2R)-2-methyl-1-pyrrolidinyl]ethyl}-1-benzofuran-5-yl)phenyl]methanone

• 常用名: cyclopropyl[4-(2-{2-[(2R)-2-methyl-1-pyrrolidinyl]ethyl}-1-benzofuran-5-yl)phenyl]methanone
• 英文名: cyclopropyl[4-(2-{2-[(2R)-2-methyl-1-pyrrolidinyl]ethyl}-1-benzofuran-5-yl)phenyl]methanone
• CAS号: 460748-73-6
• 分子量: 373.5
• 密度: N/A
• 沸点: N/A
• 分子式: C₂₅H₂₇NO₂
• 熔点: N/A
• 闪点: N/A

名称

• 英文名: cyclopropyl[4-(2-{2-[(2R)-2-methyl-1-pyrrolidinyl]ethyl}-1-benzofuran-5-yl)phenyl]methanone

物理化学性质

• 分子式: C₂₅H₂₇NO₂
• 分子量: 373.5
• InChIKey: POAWKGPFNHDXRG-QGZVFWFLSA-N
• SMILES: CC1CCCN1CCc1cc2cc(-c3ccc(C(=O)C4CC4)cc3)ccc2o1

靶点实验

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实验名称：In vitro binding affinity was determined as displacement of [3H]N-R-methylhistamine f... 来源：ChEMBL 靶标：Histamine H3 receptor External Id：CHEMBL838519

实验名称：Volume of distribution was observed in rat after intravenous administration of 1-5 mg... 来源：ChEMBL 靶标：N/A External Id：CHEMBL827268

实验名称：Half life was observed in rat after intravenous administration of 3-5 mg/kg; (n=3) 来源：ChEMBL 靶标：N/A External Id：CHEMBL839916

实验名称：In vitro binding affinity was determined as displacement of [3H]N-R-methylhistamine f... 来源：ChEMBL 靶标：Histamine H3 receptor External Id：CHEMBL828754

实验名称：Tested for its ability to block human histamine H3 receptor activation by the agonist... 来源：ChEMBL 靶标：Histamine H3 receptor External Id：CHEMBL852302

实验名称：Clearance was observed in rat after intravenous administration of 1-5 mg/kg 来源：ChEMBL 靶标：N/A External Id：CHEMBL839619

实验名称：In vitro binding affinity was determined as displacement of [3H]N-R-methylhistamine f... 来源：ChEMBL 靶标：Histamine H3 receptor External Id：CHEMBL838520

实验名称：Oral bioavailability in rat (dose 1-5 mg/kg i.v.) 来源：ChEMBL 靶标：N/A External Id：CHEMBL850993

实验名称：In vitro binding affinity was determined as displacement of [3H]N-R-methylhistamine f... 来源：ChEMBL 靶标：Histamine H3 receptor External Id：CHEMBL829004

实验名称：Concentration in brain of rats after 1 hr of intravenous administration 来源：ChEMBL 靶标：N/A External Id：CHEMBL838535

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