2-[5-Cyclohexyl-1-(2-cyclopentyl-2-oxo-ethyl)-2-oxo-1,2-dihydro-benzo[e][1,2,4]triazepin-3-yl]-N-[3-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-phenyl]-acetamide

• 常用名: 2-[5-Cyclohexyl-1-(2-cyclopentyl-2-oxo-ethyl)-2-oxo-1,2-dihydro-benzo[e][1,2,4]triazepin-3-yl]-N-[3-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-phenyl]-acetamide
• 英文名: 2-[5-Cyclohexyl-1-(2-cyclopentyl-2-oxo-ethyl)-2-oxo-1,2-dihydro-benzo[e][1,2,4]triazepin-3-yl]-N-[3-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-phenyl]-acetamide
• CAS号: 528884-77-7
• 分子量: 570.6
• 密度: N/A
• 沸点: N/A
• 分子式: C₃₁H₃₄N₆O₅
• 熔点: N/A
• 闪点: N/A

名称

• 英文名: 2-[5-Cyclohexyl-1-(2-cyclopentyl-2-oxo-ethyl)-2-oxo-1,2-dihydro-benzo[e][1,2,4]triazepin-3-yl]-N-[3-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-phenyl]-acetamide

物理化学性质

• 分子式: C₃₁H₃₄N₆O₅
• 分子量: 570.6
• InChIKey: DGKMBNVRIZTNTK-UHFFFAOYSA-N
• SMILES: C1CCC(CC1)C2=NN(C(=O)N(C3=CC=CC=C32)CC(=O)C4CCCC4)CC(=O)NC5=CC=CC(=C5)C6=NOC(=O)N6

靶点实验

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实验名称：Antagonist activity at CCK2 receptor in perfused rat stomach assessed as inhibition o... 来源：ChEMBL 靶标：Gastrin/cholecystokinin type B receptor External Id：CHEMBL889352

实验名称：Displacement of [125I]BH-CCK8-8S from CCK2 receptor in canine gastric mucosa 来源：ChEMBL 靶标：Gastrin/cholecystokinin type B receptor External Id：CHEMBL889353

实验名称：Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T... 来源：ChEMBL 靶标：Gastrin/cholecystokinin type B receptor External Id：CHEMBL889348

实验名称：Displacement of [3H]L-364718 from human recombinant CCK1 receptor expressed in CHOK1 ... 来源：ChEMBL 靶标：Cholecystokinin receptor type A External Id：CHEMBL889351

实验名称：Plasma clearance in dog at 2.5 mg/kg, iv 来源：ChEMBL 靶标：Canis lupus familiaris External Id：CHEMBL889360

实验名称：Bioavailability in po dosed dog 来源：ChEMBL 靶标：Canis lupus familiaris External Id：CHEMBL889362

实验名称：Half life beta in po dosed dog 来源：ChEMBL 靶标：Canis lupus familiaris External Id：CHEMBL889363

实验名称：Inhibition of pentagastrin-stimulated gastric acid secretion in iv dosed conscious ga... 来源：ChEMBL 靶标：Gastrin/cholecystokinin type B receptor External Id：CHEMBL889356

实验名称：Inhibition of pentagastrin-stimulated gastric acid secretion in intragastrically dose... 来源：ChEMBL 靶标：Gastrin/cholecystokinin type B receptor External Id：CHEMBL889357

实验名称：Inhibition of pentagastrin-stimulated gastric acid secretion in intraduodenal bolus d... 来源：ChEMBL 靶标：Gastrin/cholecystokinin type B receptor External Id：CHEMBL889358

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