TUG-1387

• 常用名: TUG-1387
• 英文名: TUG-1387
• CAS号: 6319-64-8
• 分子量: 315.36500
• 密度: 1.25g/cm3
• 沸点: 503.9ºC at 760 mmHg
• 分子式: C₂₁H₁₇NO₂
• 熔点: N/A
• 闪点: 258.6ºC

TUG-1387用途

TUG-1387是AH-7614和TUG-1506的类似物,在FFA4上没有活性。TUG-13087可作为评估FFA4功能的研究的阴性对照。

TUG-1387名称

• 英文名: 4-methyl-N-(9H-xanthen-9-yl)benzamide

TUG-1387生物活性

• 描述: TUG-1387是AH-7614和TUG-1506的类似物,在FFA4上没有活性。TUG-13087可作为评估FFA4功能的研究的阴性对照。
• 相关类别:
  研究领域 >> 其他
  信号通路 >> 其他 >> 其他
• 参考文献:

  [1]. Watterson KR, et al. Probe-Dependent Negative Allosteric Modulators of the Long-Chain Free Fatty Acid Receptor FFA4. Mol Pharmacol. 2017 Jun;91(6):630-641.

  [2]. Milligan G, et al. FFA4/GPR120: Pharmacology and Therapeutic Opportunities. Trends Pharmacol Sci. 2017 Sep;38(9):809-821.

TUG-1387物理化学性质

• 密度: 1.25g/cm3
• 沸点: 503.9ºC at 760 mmHg
• 分子式: C₂₁H₁₇NO₂
• 分子量: 315.36500
• 闪点: 258.6ºC
• 精确质量: 315.12600
• PSA: 38.33000
• LogP: 5.01100
• InChIKey: RWLHMQMVSKQATK-UHFFFAOYSA-N
• SMILES: Cc1ccc(C(=O)NC2c3ccccc3Oc3ccccc32)cc1
• 折射率: 1.669

TUG-1387靶点实验

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TUG-1387英文别名

• 4-methyl-N-9H-xanthen-9-yl-Benzamide
• N-xanthen-9-yl-p-toluamide
• N-(9-Xanthyl)-p-toluamid