2-(4-Acetylphenylamino)-N,N-diisopentyl-1-(3-(piperidin-1-yl)propyl)-1H-benzo[d]imidazole-6-carboxamide

• 常用名: 2-(4-Acetylphenylamino)-N,N-diisopentyl-1-(3-(piperidin-1-yl)propyl)-1H-benzo[d]imidazole-6-carboxamide
• 英文名: 2-(4-Acetylphenylamino)-N,N-diisopentyl-1-(3-(piperidin-1-yl)propyl)-1H-benzo[d]imidazole-6-carboxamide
• CAS号: 746661-28-9
• 分子量: 559.8
• 密度: N/A
• 沸点: N/A
• 分子式: C₃₄H₄₉N₅O₂
• 熔点: N/A
• 闪点: N/A

名称

• 英文名: 2-(4-Acetylphenylamino)-N,N-diisopentyl-1-(3-(piperidin-1-yl)propyl)-1H-benzo[d]imidazole-6-carboxamide

物理化学性质

• 分子式: C₃₄H₄₉N₅O₂
• 分子量: 559.8
• InChIKey: CXGYZUHRSDOJIS-UHFFFAOYSA-N
• SMILES: CC(=O)c1ccc(Nc2nc3ccc(C(=O)N(CCC(C)C)CCC(C)C)cc3n2CCCN2CCCCC2)cc1

靶点实验

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实验名称：Late-stage FRET-based cell-based primary screening assay to identify biased ligands o... 来源：The Scripps Research Institute Molecular Screening Center 靶标：melanocortin receptor 4 [Homo sapiens] External Id：MC4R_AG_FRET_384_4XEC50

实验名称：Selectivity for human MC4R over human MC3R 来源：ChEMBL 靶标：Melanocortin receptor (M3 and M4) External Id：CHEMBL896763

实验名称：Agonist activity at human melanocortin 4 receptor expressed in CHOK1 cells assessed a... 来源：ChEMBL 靶标：Melanocortin receptor 4 External Id：CHEMBL896764

实验名称：Displacement of [125I]NDP-alphaMSH from human melanocortin 5 receptor expressed in CH... 来源：ChEMBL 靶标：Melanocortin receptor 5 External Id：CHEMBL895644

实验名称：Antagonist activity at human melanocortin 4 receptor expressed in CHOK1 cells assesse... 来源：ChEMBL 靶标：Melanocortin receptor 4 External Id：CHEMBL895645

实验名称：Half life in Sprague-Dawley rat at 4.5 umol/kg, iv 来源：ChEMBL 靶标：Rattus norvegicus External Id：CHEMBL895646

实验名称：Ratio of drug level in brain to blood in Sprague-Dawley rat at 4.5 umol/kg, iv 来源：ChEMBL 靶标：N/A External Id：CHEMBL896762

实验名称：Displacement of [125I]NDP-alphaMSH from human melanocortin 4 receptor expressed in CH... 来源：ChEMBL 靶标：Melanocortin receptor 4 External Id：CHEMBL895641

实验名称：Displacement of [125I]NDP-alphaMSH from human melanocortin 1 receptor expressed in CH... 来源：ChEMBL 靶标：Melanocyte-stimulating hormone receptor External Id：CHEMBL895642

实验名称：Displacement of [125I]NDP-alphaMSH from human melanocortin 3 receptor expressed in CH... 来源：ChEMBL 靶标：Melanocortin receptor 3 External Id：CHEMBL895643

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