GPR132 antagonist 1

• 常用名: GPR132 antagonist 1
• 英文名: GPR132 antagonist 1
• CAS号: 898211-21-7
• 分子量: 359.40
• 密度: N/A
• 沸点: N/A
• 分子式: C₁₈H₁₇NO₅S
• 熔点: N/A
• 闪点: N/A

GPR132 antagonist 1用途

GPR132antagonist 1 (GPR132-B-160, 化合物 25) 是一种 GPR132 拮抗剂,EC50 值为 0.075 μM。GPR132 antagonist 1 具有促进胰岛素分泌活性,EC50值为0.7 μM。

GPR132 antagonist 1名称

• 英文名: GPR132 antagonist 1

GPR132 antagonist 1生物活性

• 描述: GPR132antagonist 1 (GPR132-B-160, 化合物 25) 是一种 GPR132 拮抗剂,EC50 值为 0.075 μM。GPR132 antagonist 1 具有促进胰岛素分泌活性,EC50值为0.7 μM。
• 相关类别:
  信号通路 >> 其他 >> 其他
  研究领域 >> 代谢疾病
• 靶点实验:

  EC50: 0.075 μM (GPR132); 0.7 μM (insulin secretion activity)[1].

• 参考文献:

  [1]. 焦宁, 等. Gpcr调节剂及其应用. 专利. CN116903563A.

GPR132 antagonist 1物理化学性质

• 分子式: C₁₈H₁₇NO₅S
• 分子量: 359.40
• InChIKey: XFMCZHXUAWBOAL-UHFFFAOYSA-N
• SMILES: Cc1c(C(=O)O)oc2ccc(S(=O)(=O)NCCc3ccccc3)cc12

GPR132 antagonist 1靶点实验

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实验名称：High-throughput screen for inhibitors of the GIV GBA-motif interaction with Galpha-i ... 来源：ICCB-Longwood/NSRB Screening Facility, Harvard Medical School External Id：HMS1303

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实验名称：AlphaScreen-based biochemical high throughput primary assay to identify activators of... 来源：The Scripps Research Institute Molecular Screening Center 靶标：N/A External Id：FBW7_ACT_ALPHA_1536_1X%ACT PRUN

实验名称：AlphaScreen-based biochemical high throughput primary assay to identify inhibitors of... 来源：The Scripps Research Institute Molecular Screening Center External Id：MITF_INH_Alpha_1536_1X%INH PRUN

实验名称：A screen for compounds that inhibit viral RNA polymerase binding and polymerization a... 来源：ICCB-Longwood/NSRB Screening Facility, Harvard Medical School 靶标：Chain A, Poliovirus Polymerase With Gtp External Id：HMS750

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