PI5P4Ks-IN-1

• 常用名: PI5P4Ks-IN-1
• 英文名: PI5P4Ks-IN-1
• CAS号: 959560-36-2
• 分子量: 331.43
• 密度: N/A
• 沸点: N/A
• 分子式: C₂₀H₁₇N₃S
• 熔点: N/A
• 闪点: N/A

PI5P4Ks-IN-1用途

PI5P4Ks-IN-1(化合物7)是一种活性化合物,对PI5P4Kα或β亚型没有检测到抑制作用[1]。

PI5P4Ks-IN-1名称

• 英文名: PI5P4Ks-IN-1

PI5P4Ks-IN-1生物活性

• 描述: PI5P4Ks-IN-1(化合物7)是一种活性化合物,对PI5P4Kα或β亚型没有检测到抑制作用[1]。
• 相关类别:
  研究领域 >> 其他
  信号通路 >> 其他 >> 其他
• 参考文献:

  [1]. Boffey HK, et al. Development of Selective Phosphatidylinositol 5-Phosphate 4-Kinase γ Inhibitors with a Non-ATP-competitive, Allosteric Binding Mode. J Med Chem. 2022;65(4):3359-3370.

PI5P4Ks-IN-1物理化学性质

• 分子式: C₂₀H₁₇N₃S
• 分子量: 331.43

PI5P4Ks-IN-1靶点实验

查看更多实验

实验名称：Inhibition of GST-fused recombinant human PI5P4Kgamma harboring insertion of QAR amin... 来源：ChEMBL 靶标：N/A External Id：CHEMBL5045802

实验名称：NCATS Kinetic Aqueous Solubility Profiling 来源：NCGC 靶标：N/A External Id：ADME-solubility1

实验名称：Primary qHTS for small molecule stabilizers of the endoplasmic reticulum resident pro... 来源：NCGC 靶标：N/A External Id：SERCaMPGLuc-p1-antagonist

实验名称：Validation qHTS for agonist of cAMP-regulated guanine nucleotide exchange factor 3 (E... 来源：NCGC External Id：epac1-activator-v

实验名称：Validation qHTS for antagonist of cAMP-regulated guanine nucleotide exchange factor 3... 来源：NCGC External Id：epac1-inhibitor-v

实验名称：Primary qHTS assay for inhibitors of alpha-synuclein gene (SNCA) expression 来源：NCGC External Id：SNCA-p-activity-luciferase

实验名称：Binding affinity to PI5P4Kgamma (unknown origin) assessed as change in melting temper... 来源：ChEMBL 靶标：Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma External Id：CHEMBL5045806

实验名称：Confirmatory qHTS assay for small molecule inhibitors of Inositol hexaphosphate kinas... 来源：NCGC External Id：IP6K1-f1-cherrypicks

实验名称：Inhibition of PI5P4Kalpha (unknown origin) by ADP-Glo assay 来源：ChEMBL 靶标：Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha External Id：CHEMBL5045805

实验名称：Validation qHTS for agonist of cAMP-regulated guanine nucleotide exchange factor 4 (E... 来源：NCGC External Id：epac2-activator-v2

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