Chinese Journal of Chemistry

A Convenient Synthesis of 2??Oxazolines and 2??Benoxazoles with PPh3??DDQ as the Dehydrating Reagent

Q Xu, Z Li, H Chen

Index: Xu, Quancai; Li, Zhengning; Chen, Huiying Chinese Journal of Chemistry, 2011 , vol. 29, # 5 p. 925 - 932

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Citation Number: 7

Abstract

Abstract 2-Oxazolines and 2-benoxazoles were synthesized in high yields from acylamino alcohols and acylamino-phenols, respectively, with triphenylphosphine-2, 3-dichloro-5, 6- dicyanobenzoquinone (PPh 3-DDQ) as the dehydrating and activating reagent. The synthesis was accomplished under neutral conditions.

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