Use of polyfunctionalized ethylene synthons: Convenient synthesis of biologically active trifluoromethyl containing N-substituted-benzoylpyrazoles and triazole

…, Z Guilong, H Fangzhong, Y Huazheng

Index: Li, Ming; Wen, Lirong; Wang, Xiao; Yao, Changsheng; Fu, Weijun; Zhao, Guilong; Hu, Fangzhong; Yang, Huazheng Indian Journal of Chemistry - Section B Organic and Medicinal Chemistry, 2006 , vol. 45, # 2 p. 483 - 488

Full Text: HTML

Citation Number: 1

Abstract

Abstract: Ten biologically active trifluoromethyl containing N-substituted-benzoylpyrazoles (3a-d, 4a-d, and 6a, b) and one triazole analogue 5 have been conveniently synthesized from four versatile polyfunctionalized ethylene synthons and one novel synthon N- cyanoimido-S, S-dimethyldithio-carbonate (CIDT, v), respectively. The reactions of trifluoromethyl containing substituted benzoylhydrazine with classical synthons such as ...