A Simple route to polysubstituted indoles exploiting azide induced furan ring opening

VT Abaev, AT Plieva, PN Chalikidi, MG Uchuskin…

Index: Hicks, Martin G.; Jones, Gurnos.; York, David C. Journal of the Chemical Society, Perkin Transactions 1: Organic and Bio-Organic Chemistry (1972-1999), 1988 , p. 69 - 76

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Citation Number: 15

Abstract

... Select a Journal or Book ... Reaction conditions: (a) for 1a–g: aldehyde 3 (10 mmol), furan 4 (22 mmol), HClO 4 (6 mmol), and 1,4-dioxane (10 mL), 5–10 °C; (b) for 1h–j: aldehyde 3 (10 mmol), furan 4 (22 mmol), Me 3 SiPPA (16.5 mmol), and CH 2 Cl 2 (10 ... 5, c, H, Cl, Ph, Me, o, 88. ...