Facile syntheses of oxazolines and thiazolines with N-acylbenzotriazoles under microwave irradiation

AR Katritzky, C Cai, K Suzuki…

Index: Journal of Organic Chemistry, , vol. 69, # 3 p. 811 - 814

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Citation Number: 106

Abstract

... The Journal of Organic Chemistry. ... Microwave reactions of 2-amino-2-methyl-1-propanol (2) or 2-aminoethanethiol hydrochloride (4) with readily available N-acylbenzotriazoles 1a−j in the presence of SOCl 2 produced 2-substituted 2-oxazolines 3a−j in 84−98% yields and 2 ...