Discovery of (R)-4-Cyclopropyl-7, 8-difluoro-5-(4-(trifluoromethyl) phenylsulfonyl)-4, 5-dihydro-1 H-pyrazolo [4, 3-c] quinoline (ELND006) and (R)-4-Cyclopropyl-8- …

G Probst, DL Aubele, S Bowers…

Index: Journal of Medicinal Chemistry, , vol. 56, # 13 p. 5261 - 5274

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Citation Number: 13

Abstract

... Journal of Medicinal Chemistry. ... Department of Medicinal Chemistry, Elan Pharmaceuticals, 180 Oyster Point ... Department of Process and Analytical Chemistry, Elan Pharmaceuticals, 180 Oyster Point Boulevard, South San Francisco, California 94080, United States. ...