Chemical Communications

Cu (I)-catalyzed intramolecular oxidative C–H amination of 2-aminoacetophenones: a convenient route toward isatins

PC Huang, P Gandeepan, CH Cheng

Index: Huang, Pang-Chi; Gandeepan, Parthasarathy; Cheng, Chien-Hong Chemical Communications, 2013 , vol. 49, # 76 p. 8540 - 8542

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Citation Number: 32

Abstract

Transition-metal-catalyzed construction of C–C and C–heteroatom bonds has become a proven method for the synthesis of bioactive compounds and advanced materials. 1 In recent years, great effort has been made toward the direct functionalization of C–H bond rather than the pre-functionalized carbon–halogen or carbon–pseudohalogen bond which requires additional steps for preparation. 2 However, most of these reactions require the ...