e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521
Syntheses and activities of new C10 β-turn peptidomimetics
…, M Pattarawarapan, S Roy, HU Saragovi…
Index: Lee, Hong Boon; Zaccaro, Maria Clara; Pattarawarapan, Mookda; Roy, Sudipta; Saragovi, H. Uri; Burgess, Kevin Journal of Organic Chemistry, 2004 , vol. 69, # 3 p. 701 - 713
A program to identify small molecules that mimic or disrupt protein-protein interactions led us to design the peptidomimetics 1-3. Solid-phase syntheses of 1-3 were developed. The purities of the crude materials isolated from the resin tend to be highest for the S-and N- compounds 2 and 3 and better than in the corresponding syntheses of peptidomimetics A. The particular dipeptide units incorporated were chosen to correspond with the turn ...