Additions of 1-(. alpha.-aminoalkyl) benzotriazoles to enol ethers. New routes to 1, 3-amino ethers

AR Katritzky, S Rachwal, B Rachwal…

Index: Katritzky, Alan R.; Rachwal, Stanislaw; Rachwal, Bogumila; Steel, Peter J. Journal of Organic Chemistry, 1992 , vol. 57, # 18 p. 4932 - 4939

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Citation Number: 24

Abstract

Center for Heterocyclic Compounds, Department of Chemistry, University of Florida, Gainesville, Florida 3261 1-2046, and Chemistry Department, University of Canterbury, New Zealand Received April 8, 1992 l-(aA min~ l) bem~ les add readily to enol ethers to give the corresponding l-benzotriazolyl-3-aminminoalkyl ethers in high yields. Subaequent replacement of the benzotriazole moiety by an alkyl or aryl group (with a Grignard reagent ...