Tetrahedron Letters

Pd-catalyzed amidation of aryl (Het) halides with tert-butyl carbamate

L Qin, H Cui, D Zou, J Li, Y Wu, Z Zhu, Y Wu

Index: Qin, Lijin; Cui, Hongmeng; Zou, Dapeng; Li, Jingya; Wu, Yangjie; Zhu, Zhiwu; Wu, Yusheng Tetrahedron Letters, 2010 , vol. 51, # 33 p. 4445 - 4448

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Citation Number: 16

Abstract

Aryl amines are traditionally valuable in organic synthesis, pharmaceuticals, and materials science. 1, 2, 3, 4 and 5 The synthesis of arylamines has always been a topic of interest in organic chemistry. 6 In the past years, palladium-catalyzed C–N coupling has received an increased attention. 7 A variety of excellent work has been carried out for this reaction. 8 Lithium bis(trimethylsilyl)amide, 8d lithium amide, 8e zinc bis(hexamethyl-disilazide), 8f and ...