Reduction of 5-(Trifluoromethyl) isoxazoles with Lithium Aluminum Hydride: Synthesis of (2, 2, 2-Trifluoroethyl) aziridines

CP Felix, N Khatimi, AJ Laurent

Index: Felix, C.; Laurent, A.; Lesniak, S.; Mison, P. Journal of Chemical Research, Miniprint, 1991 , # 2 p. 301 - 323

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Citation Number: 25

Abstract

Trifluoromethylated heterocycles are currently of considerable interest, owing to their biological potential. lS2 During our ongoing research on the synthesis of trifluoromethylated a~ iridines,~ we focused our efforts on the preparation of (2, 2, 2-trifluoroethyl) aziridines 4

~39%

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