e.g. Filippa Pettersson or Cancer Res. 75(6) , 1102-12, (2015) or 10.1002/anie.201600521

A novel three-carbon annelation method for pyridine derivatives.

金子主税，内藤俊彦，百瀬祐，下村直之…

Index: Kaneko, Chikara; Naito, Toshihiko; Momose, Yu; Shimomura, Naoyuki; Ohashi, Tetsuo; Somei, Masanori Chemical & Pharmaceutical Bulletin, 1983 , vol. 31, # 6 p. 2168 - 2171

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Citation Number: 1

Abstract

... THREE—CARBON ANNELATION METHOD FOR PYRIDINE DERIVATIVESl) Chikara Kaneko,* TOShihiko Naito, Yu Momose, Naoyuki Shimomura, Tetsuo Ohashi, and Masanori Somei Faculty of ... accessible by our two—step procedure (Kaneko—Naito method) from ...

7-(2-hydroxypropan-2-yl)-6-methoxy-3-azabicyclo[4.2.0]oct-4-en-2-one Structure

7-(2-hydroxypro...

~%

7-(2-hydroxypropan-2-yl)-3-azabicyclo[4.2.0]octa-1(6),4-dien-2-one Structure

7-(2-hydroxypro...

7-(2-hydroxypropan-2-yl)-3-azabicyclo[4.2.0]octa-1(6),4-dien-2-one Structure

7-(2-hydroxypro...

~58%

5,6-dimethyl-2,7-dihydrocyclopenta[c]pyridin-1-one Structure

5,6-dimethyl-2,...

7-(2-hydroxypropan-2-yl)-6-methoxy-3-azabicyclo[4.2.0]oct-4-en-2-one Structure

7-(2-hydroxypro...

~%

5,6-dimethyl-2,7-dihydrocyclopenta[c]pyridin-1-one Structure

5,6-dimethyl-2,...

7-(1-hydroxyethyl)-4-methyl-3-azabicyclo[4.2.0]octa-1(6),4-dien-2-one Structure

7-(1-hydroxyeth...

~45%

3,6-dimethyl-2,7-dihydrocyclopenta[c]pyridin-1-one Structure

3,6-dimethyl-2,...

7-(1-hydroxyethyl)-4-methyl-3-azabicyclo[4.2.0]octa-1(6),4-dien-2-one Structure

7-(1-hydroxyeth...

~%

3,6-dimethyl-2,5,6,7-tetrahydrocyclopenta[c]pyridin-1-one Structure

3,6-dimethyl-2,...

3,6-dimethyl-2,7-dihydrocyclopenta[c]pyridin-1-one Structure

3,6-dimethyl-2,...

~%

3,6-dimethyl-2,5,6,7-tetrahydrocyclopenta[c]pyridin-1-one Structure

3,6-dimethyl-2,...

1-(2-hydroxypropan-2-yl)-4-methyl-2,4-dihydrocyclobuta[c]quinolin-3(1H)-one Structure

1-(2-hydroxypro...

~%

1,2,5-trimethyl-3H-cyclopenta[c]quinolin-4-one Structure

1,2,5-trimethyl...

4-methyl-2,4-dihydro-3H-spiro[cyclobuta[c]quinoline-1,2'-oxiran]-3-one Structure

4-methyl-2,4-di...

~%

5-methyl-2,3-dihydrocyclopenta[c]quinoline-1,4-dione Structure

5-methyl-2,3-di...

4-methyl-1-methylidene-2H-cyclobuta[c]quinolin-3-one Structure

4-methyl-1-meth...

~%

5-methyl-2,3-dihydrocyclopenta[c]quinoline-1,4-dione Structure

5-methyl-2,3-di...

8b-methoxy-4-methyl-1-methylene-1,2,2a,8b-tetrahydrocyclobuta(c)quinolin-3(4H)-one Structure

8b-methoxy-4-me...

~%

5-methyl-2,3-dihydrocyclopenta[c]quinoline-1,4-dione Structure

5-methyl-2,3-di...

1-Dimethoxymethyl-4-methyl-2,4-dihydro-1H-cyclobuta[c]quinolin-3-one Structure

1-Dimethoxymeth...

~12%

5-methyl-1,3-dihydrocyclopenta[c]quinoline-2,4-dione Structure

5-methyl-1,3-di...