Antimalarial activity enhancement in hydroxymethylcarbonyl (HMC) isostere-based dipeptidomimetics targeting malarial aspartic protease plasmepsin

K Hidaka, T Kimura, AJ Ruben, T Uemura…

Index: Bioorganic and Medicinal Chemistry, , vol. 16, # 23 p. 10049 - 10060

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Citation Number: 30

Abstract

... Bioorganic & Medicinal Chemistry. ... for Frontier Research in Medicinal Science, 21st Century COE Program, Kyoto Pharmaceutical University, Yamashina-ku ... Institute, Johns Hopkins University, Baltimore, MD 21218, USA; c Department of Medicinal Chemistry, Tokyo University of ...