Synthesis and radiosynthesis with a positron emitter of EP 00652218, a potent antagonist of NK1 receptor, and of a fluoro analog for in vivo evaluation of the …

C Gueret, MD Le Bas, C Perrio…

Index: Journal of Labelled Compounds and Radiopharmaceuticals, , vol. 44, p. S283 - S285

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Citation Number: 4

Abstract

... In this paper we report both the synthesis and labelling of the reference EP 00652218 1 with carbon-1 1 and of the ... 5a and 5b were then transformed into the bromo 6a,7a and chloro 6b compounds respectively, according to a described procedure ... J. Labelled Cpd Radiophann. ...