A novel, high-affinity, fluorescent progesterone receptor antagonist. Synthesis and in vitro studies

C Hödl, WSL Strauss, R Sailer, C Seger…

Index: Acosta, Kirk; Cessac, James W.; Rao, P. Narasimha; Kim, Hyun K. Journal of the Chemical Society, Chemical Communications, 1994 , # 17 p. 1985 - 1986

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Citation Number: 14

Abstract

... 2.760 mmol) were dissolved in anhydrous DMF (4.0 mL) and stirred in the presence of dry K 2 CO 3 ... IR (KBr): 3430 (s, O−H); 2934 (m, C−H); 2861 (m, C−H); 1737 (w, C O ... After thawing cells were incubated with 50 μL p-nitrophenyl phosphate (5 mM, Fluka) dissolved in aqueous ...