Arkivoc

A new protocol for the synthesis of primary, secondary and tertiary anthranilamides utilizing N-(2-aminoarylacyl) benzotriazoles

N Kanışkan, Ş Kökten, İ Çelik

Index: Kaniskan, Nevin; Koekten, Sule; Celik, Ilhami Arkivoc, 2012 , vol. 2012, # 8 p. 198 - 213

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Citation Number: 5

Abstract

Abstract A convenient route for efficient conversion of unprotected anthranilic acids into the corresponding N-(2-aminoarylacyl) benzotrazoles is described. N-(2-Aminoarylacyl)- benzotrazoles have been successfully used to synthesize primary, secondary and tertiary anthranilamides in high yields (71-96%). Keywords: Anthranilic acid, benzotriazole, N-(2- aminoarylacyl) benzotrazoles, anthranilamides