High-affinity and potent, water-soluble 5-amino-1, 4-benzodiazepine CCKB/gastrin receptor antagonists containing a cationic solubilizing group

GA Showell, S Bourrain, JG Neduvelil…

Index: Journal of Medicinal Chemistry, , vol. 37, # 6 p. 719 - 721

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Citation Number: 69

Abstract

... The electron-withdrawing nature of the carbamate group may activate the double bond to hydrogenation and subsequently the NO bond to hy- 0022-2623/94/1837-0719$04.50/0 0 1994 American Chemical Society ... 720 Journal of Medicinal Chemistry, 1994, Vol. ...